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Belzutifan (PT2977)

Product Specifications

CAS Number

1672668-24-4

Synonyms

MK-6482

Target

HIF

Applications

Angiogenesis

Smiles

CS (=O) (=O) C1=C2C (C (C (C2=C (C=C1) OC3=CC (=CC (=C3) C#N) F) F) F) O

Molecular Formula

C17H12F3NO4S

Additionnal Information

Belzutifan (PT2977), an orally active and selective HIF-2α inhibitor, increases potency and improves pharmacokinetic profile, providing a potential treatment for clear cell renal cell carcinoma (ccRCC) .

Storage Conditions

3 years -20°C powder

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