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ODM-203

Product Specifications

CAS Number

1430723-35-5

Target

FGFR

Applications

Protein Tyrosine Kinase

Smiles

CN1C=C (C=N1) C2=CC3=C (C=C2) N (C=N3) C4=CC (=CC (=C4) NS (=O) (=O) C5CC5) C6=C (C=C (C=C6) F) F

Molecular Formula

C26H21F2N5O2S

Additionnal Information

ODM-203 is a selective inhibitor of FGFR and VEGFR with ic50s of 11 nM,16 nM,6 nM, 35 nM,26 nM,9 nM,5 nM for recombinant FGFR1, FGFR2, FGFR3, FGFR4, VEGFR1, VEGFR2 and VEGFR3, respectively.

Storage Conditions

3 years -20°C powder

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