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GSK8612

Product Specifications

CAS Number

2361659-62-1

Target

TBK1

Applications

Immunology & Inflammation

Smiles

CC1=NN (C=C1NC2=NC=C (C (=N2) NCC3=CC=C (C=C3) S (=O) (=O) N) Br) CC (F) (F) F

Molecular Formula

C17H17BrF3N7O2S

Additionnal Information

GSK8612 is a highly potent and selective inhibitor for TBK1 (Tank-binding Kinase-1) with pKd of 8.0. Within 10-fold affinity with respect to TBK1, no off-targets of GSK8612 could be identified.

Storage Conditions

3 years -20°C powder

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