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GSK3368715 3HCl

Product Specifications

CAS Number

2227587-26-8

Synonyms

EPZ019997 3HCl

Target

PRMT

Applications

Epigenetics

Smiles

Cl.Cl.Cl.CCOCC1 (CCC (CC1) C2=N[NH]C=C2CN (C) CCNC) COCC

Molecular Formula

C20H41Cl3N4O2

Additionnal Information

GSK3368715 3HCl is a potent inhibitor of type I protein arginine methyltransferases (PRMT) that inhibits PRMT1, 3, 4, 6 and 8 with Kiapp vaules ranging from 1.5 to 81 nM.

Storage Conditions

3 years -20°C powder

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