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MRTX-1257

Product Specifications

CAS Number

2206736-04-9

Target

Ras

Applications

Apoptosis

Molecular Formula

C33H39N7O2

Additionnal Information

MRTX-1257 is a potent, selective, irreversible, covalent and orally active inhibitor of KRAS G12C with IC50 of 900 pM for KRAS dependent ERK phosphorylation in H358 cells.

Storage Conditions

3 years -20°C powder

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