What is the catalog number for Ripretinib?

The catalog number for Ripretinib is S8757-100mg.

What sizes are available for Ripretinib?

Ripretinib is available in the following size(s): 100 mg.

Is Ripretinib in stock?

Ripretinib is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures Ripretinib?

Ripretinib is manufactured by Bimake.

What is the estimated delivery time for Ripretinib?

Estimated delivery time for Ripretinib is approximately 15 business day(s), depending on your location.

Ripretinib

Product Specifications

CAS Number

1442472-39-0

Synonyms

DCC-2618

Target

C-Kit

Applications

Protein Tyrosine Kinase

Smiles

CCN1C2=CC (=NC=C2C=C (C1=O) C3=CC (=C (C=C3Br) F) NC (=O) NC4=CC=CC=C4) NC

Molecular Formula

C24H21BrFN5O2

Additionnal Information

Ripretinib is an orally bioavailable switch pocket control inhibitor of wild-type and mutated forms of the tumor-associated antigens (TAA) mast/stem cell factor receptor (SCFR) Kit (c-Kit) and PDGFR-alpha, with IC50 values of 4 nM, 8 nM, 18 nM, 5 nM and 14 nM for WT Kit (c-Kit), V654A Kit (c-Kit), T670I Kit (c-Kit), D816H Kit (c-Kit) and D816V Kit (c-Kit), respectively.