Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

Tropifexor (LJN452)

Product Specifications

CAS Number

1383816-29-2

Target

FXR

Applications

Metabolism

Smiles

C1CC1C2=C (C (=NO2) C3=CC=CC=C3OC (F) (F) F) COC4CC5CCC (C4) N5C6=NC7=C (C=C (C=C7S6) C (=O) O) F

Molecular Formula

C29H25F4N3O5S

Additionnal Information

Tropifexor (LJN452) is a novel and highly potent agonist of FXR with EC50 of 0.2 nM in HTRF assay. It shows no significant off-target activity against a broad panel of enzyme, ion channel, nuclear receptor, and GPCR (>10000-fold selectivity for FXR) .

Storage Conditions

3 years -20°C powder

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Ethyl Caproate
TRC-E901600-50G 50 g

Ethyl Caproate

Sign In for Pricing
View Details
Tissue FFPE Sections, Myeloid tissue
CS808511 5x 5 µm

Tissue FFPE Sections, Myeloid tissue

Sign In for Pricing
View Details
IgM Immunoglobulin (Cocktail), CF488A conjugate, 0.1mg/mL
BNC880762-100 1x 100 µL

IgM Immunoglobulin (Cocktail), CF488A conjugate, 0.1mg/mL

Sign In for Pricing
View Details
NABP1 Mouse Monoclonal Antibody [Clone ID: OTI7D9]
CF811089 100 µg

NABP1 Mouse Monoclonal Antibody [Clone ID: OTI7D9]

Sign In for Pricing
View Details
p16INK4A (CDKN2A) Mouse Monoclonal Antibody (HRP conjugated) [Clone ID: OTI4E9]
TA805241BM 100 µL

p16INK4A (CDKN2A) Mouse Monoclonal Antibody (HRP conjugated) [Clone ID: OTI4E9]

Sign In for Pricing
View Details
Collagen VI Recombinant Rabbit monoclonal Antibody
HA750305 100 µL

Collagen VI Recombinant Rabbit monoclonal Antibody

Sign In for Pricing
View Details