Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

Nemtabrutinib (ARQ 531)

Product Specifications

CAS Number

2095393-15-8

Synonyms

MK-1026

Target

BTK

Applications

Protein Tyrosine Kinase

Smiles

C1CC (OCC1NC2=NC=NC3=C2C (=CN3) C (=O) C4=C (C=C (C=C4) OC5=CC=CC=C5) Cl) CO

Molecular Formula

C25H23ClN4O4

Additionnal Information

Nemtabrutinib (ARQ 531, MK-1026) is an ATP-competitive tyrosine kinase inhibitor designed to target BTK with an IC50 of 0.85 nM. It also has a distinct kinase selectivity profile with strong inhibitory activity against several key oncogenic drivers from TEC, Trk and Src family kinases.

Storage Conditions

3 years -20°C powder

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

NF-kappaB p105/p50 Conjugated Antibody
MBS9455879-01 0.1 mL (Biotin)

NF-kappaB p105/p50 Conjugated Antibody

Sign In for Pricing
View Details
NF-kappaB p105/p50 Conjugated Antibody
MBS9455879-02 0.1 mL (AF350)

NF-kappaB p105/p50 Conjugated Antibody

Sign In for Pricing
View Details
NF-kappaB p105/p50 Conjugated Antibody
MBS9455879-03 0.1 mL (AF405)

NF-kappaB p105/p50 Conjugated Antibody

Sign In for Pricing
View Details
NF-kappaB p105/p50 Conjugated Antibody
MBS9455879-04 0.1 mL (AF488)

NF-kappaB p105/p50 Conjugated Antibody

Sign In for Pricing
View Details
NF-kappaB p105/p50 Conjugated Antibody
MBS9455879-05 0.1 mL (AF555)

NF-kappaB p105/p50 Conjugated Antibody

Sign In for Pricing
View Details
NF-kappaB p105/p50 Conjugated Antibody
MBS9455879-06 0.1 mL (AF594)

NF-kappaB p105/p50 Conjugated Antibody

Sign In for Pricing
View Details