What is the catalog number for Theliatinib (HMPL-309)?

The catalog number for Theliatinib (HMPL-309) is S8584-5mg.

What sizes are available for Theliatinib (HMPL-309)?

Theliatinib (HMPL-309) is available in the following size(s): 5 mg.

Is Theliatinib (HMPL-309) in stock?

Theliatinib (HMPL-309) is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures Theliatinib (HMPL-309)?

Theliatinib (HMPL-309) is manufactured by Bimake.

What is the estimated delivery time for Theliatinib (HMPL-309)?

Estimated delivery time for Theliatinib (HMPL-309) is approximately 15 business day(s), depending on your location.

Theliatinib (HMPL-309)

Product Specifications

CAS Number

1353644-70-8

Target

EGFR

Applications

Protein Tyrosine Kinase

Smiles

COC1=C (NC (=O) N2CC3CCN (C) C3C2) C=C4C (=NC=NC4=C1) NC5=CC (=CC=C5) C#C

Molecular Formula

C25H26N6O2

Additionnal Information

Theliatinib (HMPL-309) is a highly potent EGFR inhibitor with Ki value of 0.05 nM against the wild type EGFR and IC50 values of 3 nM and 22 nM against EGFR and EGFR T790M/L858R mutant. It demonstrats 50 fold greater selectivity for EGFR compared to 72 other kinases.