ARV-771
Product Specifications
CAS Number
1949837-12-0
Target
PROTAC
Applications
Others
Smiles
CC1=C (SC2=C1C (=NC (C3=NN=C (N32) C) CC (=O) NCCOCCCOCC (=O) NC (C (=O) N4CC (CC4C (=O) NC (C) C5=CC=C (C=C5) C6=C (N=CS6) C) O) C (C) (C) C) C7=CC=C (C=C7) Cl) C
Molecular Formula
C49H60ClN9O7S2
Additionnal Information
ARV-771 is a potent pan- (bromodomain and extra-terminal) BET degrader, a novel BET-PROTAC (proteolysis-targeting chimera) with Kd of 34 nM, 4.7 nM, 8.3 nM, 7.6 nM, 9.6 nM, and 7.6 nM for BRD2 (1), BRD2 (2), BRD3 (1), BRD3 (2), BRD4 (1), and BRD4 (2), respectively.
Storage Conditions
3 years -20°C powder
More Discoveries
Explore Other Products
Browse additional items from our catalog
UEB17182-01 250 mg
5,6,7,8-Tetrahydroimidazo[1,2-a]pyridine-6-carboxylic Acid hydrochloride
Sign In for Pricing
View Details