Trilaciclib
Product Specifications
CAS Number
1374743-00-6
Synonyms
G1T28, G1T28-1
Target
CDK
Applications
Cell Cycle
Smiles
CN1CCN (CC1) C2=CN=C (C=C2) NC3=NC=C4C=C5C (=O) NCC6 (N5C4=N3) CCCCC6
Molecular Formula
C24H30N8O
Additionnal Information
Trilaciclib is a highly potent, selective and reversible cyclin-dependent kinase 4 and 6 (CDK4/6) inhibitor. Trilaciclib inhibits CDK4/cyclin D1 and CDK6/cyclin D3 with IC50 of 1 nM and 4 nM, respectively.
Storage Conditions
3 years -20°C powder
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