PF-4136309

857679-55-1

INCB8761, PF-04136309

CCR

GPCR & G Protein

OC1 (CCC (CC1) NC2CCN (C2) C (=O) CNC (=O) C3=CC (=CC=C3) C (F) (F) F) C4=NC=C (C=C4) C5=NC=CC=N5

C29H31F3N6O3

PF-4136309 (INCB8761, PF-04136309) is a potent, selective, and orally bioavailable CCR2 antagonist with an IC50 of 5.2 nM for human CCR2.

3 years -20°C powder