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PT2399

Product Specifications

CAS Number

1672662-14-4

Target

HIF

Applications

Angiogenesis

Smiles

C1C2=C (C=CC (=C2C (C1 (F) F) O) S (=O) (=O) C (F) F) OC3=CC (=CC (=C3) C#N) F

Molecular Formula

C17H10F5NO4S

Additionnal Information

PT2399 is a potent and orally available antagonist of HIF-2 that selectively disrupts the heterodimerization of HIF-2α with HIF-1β.

Storage Conditions

3 years -20°C powder

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