RapaLink-1
Product Specifications
CAS Number
1887095-82-0
Target
MTOR
Applications
PI3K/Akt/mTOR
Molecular Formula
C91H138N12O24
Additionnal Information
RapaLink-1, a third-generation bivalent inhibitor of mTOR, combines Rapamycin with MLN0128 using an inert chemical linker. It demonstrates efficacy against resistant mutants of malignant brain tumors and inhibits cancer cell progression by binding to mesenchymal markers.
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