Pelabresib (CPI-0610)
Product Specifications
CAS Number
1380087-89-7
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
CC1=NOC2=C1C3=CC=CC=C3C (=NC2CC (=O) N) C4=CC=C (C=C4) Cl
Molecular Formula
C20H16ClN3O2
Additionnal Information
Pelabresib (CPI-0610) is a potent and selective benzoisoxazoloazepine BET bromodomain inhibitor with an IC50 of 39 nM for BRD4-BD1 in TR-FRET assay and currently undergoing human clinical trials for hematological malignancies. CPI-0610 inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes.
Storage Conditions
2 years -80 in solvent
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