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GSK199

Product Specifications

CAS Number

1549811-53-1

Target

PAD

Applications

Metabolism

Molecular Formula

C24H28N6O2.ClH

Additionnal Information

GSK199 is a reversible, specific inhibitor of peptidyl arginine deiminase 4 (PAD4), with an IC50 of 200 nM without calcium. It is involved in histone citrullination and neutrophil extracellular trap formation, making it useful for studying autoimmune, cardiovascular, and oncological diseases.

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