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Akti-1/2

Product Specifications

CAS Number

612847-09-3

Synonyms

Akt Inhibitor VIII

Target

Akt

Applications

PI3K/Akt/mTOR

Smiles

C1CN (CCC1N2C3=CC=CC=C3NC2=O) CC4=CC=C (C=C4) C5=C (N=C6C=C7C (=NC=N7) C=C6N5) C8=CC=CC=C8

Molecular Formula

C34H29N7O

Additionnal Information

Akti-1/2 (Akt Inhibitor VIII) is a highly selective Akt1/Akt2 inhibitor with IC50 of 58 nM/210 nM, respectively, about 36-fold selectivity for Akt1 over Akt3. Akti-1/2 induces apoptosis.

Storage Conditions

2 years -80 in solvent

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