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Defactinib (VS-6063)

Product Specifications

CAS Number

1073154-85-4

Synonyms

PF-04554878

Target

FAK

Applications

Protein Tyrosine Kinase

Smiles

CNC (=O) C1=CC=C (C=C1) NC2=NC=C (C (=N2) NCC3=NC=CN=C3N (C) S (=O) (=O) C) C (F) (F) F

Molecular Formula

C20H21F3N8O3S

Additionnal Information

Defactinib (VS-6063, PF-04554878) is a selective, and orally active FAK inhibitor. Phase 2.

Storage Conditions

2 years -80 in solvent

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