MS417
Product Specifications
CAS Number
916489-36-6
Synonyms
GTPL7512
Target
Epigenetic Reader Domain
Applications
Epigenetics
Molecular Formula
C20H19ClN4O2S
Additionnal Information
MS417 is a selective BET-specific BRD4 inhibitor, binds to BRD4-BD1 and BRD4-BD2 with IC50s of 30, 46 nM and Kds of 36.1, 25.4 nM, respectively, with weak selectivity at CBP BRD (IC50, 32.7 μM) .
More Discoveries
Explore Other Products
Browse additional items from our catalog