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MS417

Product Specifications

CAS Number

916489-36-6

Synonyms

GTPL7512

Target

Epigenetic Reader Domain

Applications

Epigenetics

Molecular Formula

C20H19ClN4O2S

Additionnal Information

MS417 is a selective BET-specific BRD4 inhibitor, binds to BRD4-BD1 and BRD4-BD2 with IC50s of 30, 46 nM and Kds of 36.1, 25.4 nM, respectively, with weak selectivity at CBP BRD (IC50, 32.7 μM) .
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