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GSK-LSD1 2HCl

Product Specifications

CAS Number

2102933-95-7

Target

Histone Demethylase

Applications

Epigenetics

Smiles

C1CNCCC1NC2CC2C3=CC=CC=C3.Cl.Cl

Molecular Formula

C14H22Cl2N2

Additionnal Information

GSK-LSD1 2HCl is an irreversible, and selective LSD1 inhibitor with IC50 of 16 nM, > 1000 fold selective over other closely related FAD utilizing enzymes (i.e. LSD2, MAO-A, MAO-B) .

Storage Conditions

2 years -80 in solvent

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