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AMG 925

Product Specifications

CAS Number

1401033-86-0

Target

FLT3

Applications

Protein Tyrosine Kinase

Smiles

CC1CCC (CC1) N2C3=C (C=CN=C3) C4=CN=C (N=C42) NC5=NC6=C (CN (CC6) C (=O) CO) C=C5

Molecular Formula

C26H29N7O2

Additionnal Information

AMG 925 is a potent and orally bioavailable dual FLT3/CDK4 inhibitor with IC50 of 1 nM and 3 nM, respectively.

Storage Conditions

2 years -80 in solvent

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