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MPI-0479605

Product Specifications

CAS Number

1246529-32-7

Target

MPS1

Applications

Cytoskeletal Signaling

Smiles

CC1=C (C=CC (=C1) N2CCOCC2) NC3=NC4=C (C (=N3) NC5CCCCC5) NC=N4

Molecular Formula

C22H29N7O

Additionnal Information

MPI-0479605 is an ATP competitive and selective inhibitor of mitotic kinase Mps1 with IC50 of 1.8 nM, >40-fold selectivity over other kinases.

Storage Conditions

2 years -80 in solvent

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