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NU9056

Product Specifications

CAS Number

1450644-28-6

Target

Histone Acetyltransferase

Applications

Epigenetics

Molecular Formula

C6H4N2S4

Additionnal Information

NU9056 is a potent and selective inhibitor of Tip60 (KAT5) histone acetyltransferase with an IC50 value of 2 μM. NU9056 demonstrates over 16-fold selectivity for Tip60 compared to PCAF, p300, and GCN5 and effectively induces apoptosis in prostate cancer cells.

Storage Conditions

2 years -20°C liquid

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