Apabetalone (RVX-208)
Product Specifications
CAS Number
1044870-39-4
Synonyms
RVX-000222
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
CC1=CC (=CC (=C1OCCO) C) C2=NC3=C (C (=CC (=C3) OC) OC) C (=O) N2
Molecular Formula
C20H22N2O5
Additionnal Information
Apabetalone (RVX-208, RVX-000222) is a potent BET bromodomain inhibitor with IC50 of 0.510 μM for BD2 in a cell-free assay, about 170-fold selectivity over BD1. Phase 2.
Storage Conditions
2 years -80 in solvent
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
LC428450 20 µg
WDR79 (WRAP53) (NM_001143990) Human Over-expression Lysate
Sign In for Pricing
View Details TP300097 20 µg
Apc11 (ANAPC11) (NM_001002244) Human Recombinant Protein
Sign In for Pricing
View Details 
MBS1882570-01 100 Tests
PE-conjugated Anti-CEACAM5 antibody (DM122); Rabbit mAb
Sign In for Pricing
View Details MBS1882570-02 5x 100 Tests
PE-conjugated Anti-CEACAM5 antibody (DM122); Rabbit mAb
Sign In for Pricing
View Details