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Crenigacestat (LY3039478)

Product Specifications

CAS Number

1421438-81-4

Target

Notch

Applications

Neuronal Signaling

Smiles

CC (C (=O) NC1C2=CC=CC=C2C3=C (N=CC=C3) N (C1=O) CCO) NC (=O) CCC (F) (F) F

Molecular Formula

C22H23F3N4O4

Additionnal Information

Crenigacestat (LY3039478) is an oral Notch and gamma-secretase inhibitor with IC50 of 0.41 nM for Notch.

Storage Conditions

2 years -80 in solvent

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