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DMH1

Product Specifications

CAS Number

1206711-16-1

Target

TGF-beta/Smad

Applications

TGF-beta/Smad

Smiles

CC (C) OC1=CC=C (C=C1) C2=CN3C (=C (C=N3) C4=CC=NC5=CC=CC=C45) N=C2

Molecular Formula

C24 H20 N4 O

Additionnal Information

DMH1 is a selective BMP receptor inhibitor with IC50 of 107.9 nM for ALK2, exhibiting no inhibition on AMPK, ALK5, KDR (VEGFR-2) or PDGFR. DMH1 inhibits autophagy.

Storage Conditions

2 years -80 in solvent

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