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GW284543 (UNC10225170)

Product Specifications

CAS Number

790186-68-4

Target

MEK

Applications

Protein Tyrosine Kinase

Smiles

COC1=CC2=C (C=C1OC) C (=CC=N2) NC3=CC (=CC=C3) OC4=CC=CC=C4

Molecular Formula

C23H20N2O3

Additionnal Information

GW284543 (UNC10225170), a MEK5-selective inhibitor, inhibits MEK5 in a dose-dependently way as determined by reductions in pERK5, and decreases endogenous MYC protein.

Storage Conditions

3 years -20°C powder

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