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GK921

Product Specifications

CAS Number

1025015-40-0

Target

Glutaminase

Applications

Proteases

Smiles

C1CCN (C1) CCOC2=NC3=C (N=CC=C3) N=C2C#CC4=CC=CC=C4

Molecular Formula

C21H20N4O

Additionnal Information

GK921 is a transglutaminase 2 (TGase 2) inhibitor with an IC50 of 8.93 μM under a modified assay condition.

Storage Conditions

3 years -20°C powder

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