I-BET151 (GSK1210151A)
Product Specifications
CAS Number
1300031-49-5
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
CC1=C (C (=NO1) C) C2=C (C=C3C (=C2) N=CC4=C3N (C (=O) N4) C (C) C5=CC=CC=N5) OC
Molecular Formula
C23H21N5O3
Additionnal Information
I-BET151 (GSK1210151A) is a novel selective BET inhibitor for BRD2, BRD3 and BRD4 with IC50 of 0.5 μM, 0.25 μM, and 0.79 μM in cell-free assays, respectively.
Storage Conditions
2 years -80 in solvent
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