VU0238429
Product Specifications
CAS Number
1160247-92-6
Synonyms
M5 PAM
Target
AChR
Applications
Neuronal Signaling
Smiles
COC1=CC=C (C=C1) CN2C3=C (C=C (C=C3) OC (F) (F) F) C (=O) C2=O
Molecular Formula
C17H12F3NO4
Additionnal Information
VU0238429 (M5 PAM) is the first positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5/M5) with EC50 of 1.16 μM at M5 and both > 30 μM at M1 and M3. VU0238429 shows no potentiator activity at M2 or M4.
Storage Conditions
3 years -20°C powder
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