Tolvaptan

150683-30-0

OPC-41061

Vasopressin Receptor

GPCR & G Protein

CC1=CC=CC=C1C (=O) NC2=CC (=C (C=C2) C (=O) N3CCCC (C4=C3C=CC (=C4) Cl) O) C

C26H25ClN2O3

Tolvaptan (OPC-41061) is an orally effective nonpeptide arginine vasopressin V2 receptor antagonist with IC50 of 3 nM, used to treat hyponatremia.

2 years -80 in solvent