Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

Momelotinib (CYT387)

Product Specifications

CAS Number

1056634-68-4

Synonyms

LM-1149 , CYT11387

Target

JAK

Applications

Angiogenesis

Smiles

C1COCCN1C2=CC=C (C=C2) NC3=NC=CC (=N3) C4=CC=C (C=C4) C (=O) NCC#N

Molecular Formula

C23H22N6O2

Additionnal Information

Momelotinib (CYT387, LM-1149 , CYT11387) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50 of 11 nM/18 nM, ~10-fold selectivity versus JAK3. Momelotinib (CYT387) induces apoptosis and autophagy. Phase 3.

Storage Conditions

3 years -20°C (in the dark) powder

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Recombinant Human HMGB1, His-tag
P7163-100μg 100 µg

Recombinant Human HMGB1, His-tag

Sign In for Pricing
View Details
RBM14 Antibody - C-terminal region
OAAB07799-400UL 400 µL

RBM14 Antibody - C-terminal region

Sign In for Pricing
View Details
EBV-LMP1 (EBV Latent Membrane Protein 1) discontinued
376311 500 µg

EBV-LMP1 (EBV Latent Membrane Protein 1) discontinued

Sign In for Pricing
View Details
STF-083010
CST 92208S 5 mg

STF-083010

Sign In for Pricing
View Details
(±) -ANAP
HY-101937A 1 Each

(±) -ANAP

Sign In for Pricing
View Details
Recombinant Human RANK L/TRANCE/TNFSF11/CD254 Protein
RP00928 10 µg

Recombinant Human RANK L/TRANCE/TNFSF11/CD254 Protein

Sign In for Pricing
View Details