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A-966492

Product Specifications

CAS Number

934162-61-5

Target

PARP

Applications

DNA Damage/DNA Repair

Smiles

C1CC (NC1) C2=CC (=C (C=C2) C3=NC4=C (C=CC=C4N3) C (=O) N) F

Molecular Formula

C18H17FN4O

Additionnal Information

A-966492 is a novel and potent inhibitor of PARP1 and PARP2 with Ki of 1 nM and 1.5 nM, respectively.

Storage Conditions

2 years -80 in solvent

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