PFI-1 (PF-6405761)
Product Specifications
CAS Number
1403764-72-6
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
CN1CC2=C (C=CC (=C2) NS (=O) (=O) C3=CC=CC=C3OC) NC1=O
Molecular Formula
C16H17N3O4S
Additionnal Information
PFI-1 (PF-6405761) is a highly selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 μM and for BRD2 with IC50 of 98 nM in a cell-free assay.
Storage Conditions
2 years -80 in solvent
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