What is the catalog number for RP-64477?

The catalog number for RP-64477 is S0820-25mg.

What sizes are available for RP-64477?

RP-64477 is available in the following size(s): 25 mg.

Is RP-64477 in stock?

RP-64477 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures RP-64477?

RP-64477 is manufactured by Bimake.

What is the estimated delivery time for RP-64477?

Estimated delivery time for RP-64477 is approximately 15 business day(s), depending on your location.

RP-64477

Product Specifications

CAS Number

135239-65-5

Target

Acyltransferase

Applications

Metabolism

Smiles

CCCCCCCCCCOC1=CC=C (C=C1) C (=O) NC2=C (C=CC (=C2) C (=O) NCCCC) SC

Molecular Formula

C29H42N2O3S

Additionnal Information

RP-64477 is a potent inhibitor of the cholesterol esterifying enzyme Acyl-coenzyme A:cholesterol O-acyltransferase (ACAT) . RP-64477 inhibits ACAT activity with IC50 of 113 nM, 503 nM, and 180 nM in human intestinal (CaCo-2), hepatic (HepG2) and monocytic (THP-1) cell assays, respectively.