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GeA-69

Product Specifications

CAS Number

2143475-98-1

Target

PARP

Applications

DNA Damage/DNA Repair

Smiles

CC (=O) NC1=CC=CC=C1C2=CC=CC3=C2NC4=CC=CC=C34

Molecular Formula

C20H16N2O

Additionnal Information

GeA-69 is a cell-permeable, selective allosteric inhibitor targeting macrodomain 2 (MD2) of poly-adenosine-diphosphate-ribose polymerase 14 (PARP14) with Kd of 860 nM.

Storage Conditions

3 years -20°C powder

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