XCT790
Product Specifications
CAS Number
725247-18-7
Synonyms
Compound 12
Target
Estrogen/progestogen Receptor
Applications
Endocrinology & Hormones
Smiles
COC1=C (C=CC (=C1) C=C (C#N) C (=O) NC2=NN=C (S2) C (F) (F) F) OCC3=C (C=C (C=C3) C (F) (F) F) C (F) (F) F
Molecular Formula
C23H13F9N4O3S
Additionnal Information
XCT-790 (Compound 12) is a potent and selective inverse agonist for estrogen-related receptor α (ERRα) with IC50 of 0.37 μM. XCT-790 (Compound 12) is inactive against ERRγ and the estrogen receptors ERα and ERβ. XCT-790 (Compound 12) significantly inhibits in vivo tumor growth and angiogenesis, and induces apoptosis.
Storage Conditions
3 years -20°C powder
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