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GSK4716

Product Specifications

CAS Number

101574-65-6

Target

Estrogen/progestogen Receptor

Applications

Endocrinology & Hormones

Smiles

CC (C) C1=CC=C (C=C1) C=NNC (=O) C2=CC=C (C=C2) O

Molecular Formula

C17H18N2O2

Additionnal Information

GSK4716 is a selective agonist of Estrogen-Related Orphan Nuclear Receptors ERR and ERRγ with an IC50 of 2 μM in the ERRγ FRET assay.

Storage Conditions

3 years -20°C powder

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