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Amezalpat

Product Specifications

CAS Number

1616372-41-8

Synonyms

TPST-1120

Additionnal Information

Amezalpat is a first-in-class, oral, competitive antagonist of peroxisome proliferator-activated receptor α (PPARα), with IC50 of 0.04 μM. It inhibits fatty acid oxidation (FAO), disrupting cancer cell metabolism and restoring immune responses, and shows antitumor activity in research on advanced solid tumors.

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