RJG-2051
Product Specifications
CAS Number
2851993-77-4
Target
AKR1C
Applications
Immunology & Inflammation
Additionnal Information
RJG-2051 is a selective covalent SuTEx inhibitor of AKR1C3 with an IC50 of 13 nM that targets a noncatalytic tyrosine residue (Y24), effectively blocking its enzymatic activity and disrupting androgen, estrogen, and prostaglandin metabolism.
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