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RJG-2051

Product Specifications

CAS Number

2851993-77-4

Target

AKR1C

Applications

Immunology & Inflammation

Additionnal Information

RJG-2051 is a selective covalent SuTEx inhibitor of AKR1C3 with an IC50 of 13 nM that targets a noncatalytic tyrosine residue (Y24), effectively blocking its enzymatic activity and disrupting androgen, estrogen, and prostaglandin metabolism.

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