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GS-6201

Product Specifications

CAS Number

752222-83-6

Synonyms

CVT-6883

Additionnal Information

GS-6201 (CVT-6883) is a selective adenosine A2B receptor antagonist. GS-6201 displays high affinity and selectivity for the human adenosine A2B receptors (Ki=22 nM) . GS-6201 reduces caspase-1 activity in the heart, and attenuates cardiac remodeling after acute myocardial infarction (AMI) in the mouse. GS-62013 attenuates the airway reactivity induced by NECA, AMP, or allergen in sensitized mice.

Storage Conditions

3 years-20°C powder 2 years-80°C in solvent

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