CP-100356 hydrochloride
Product Specifications
CAS Number
142715-48-8
Target
BCRP
Applications
Transmembrane Transporters
Molecular Formula
C31H36N4O6.ClH
Additionnal Information
CP-100356 hydrochloride is an orally active dual inhibitor of MDR1 (P-gp) and BCRP, with IC50 of ∼0.5 μM for MDR1-mediated calcein-AM transport inhibition and ∼1.5 μM for BCRP-mediated prazosin transport inhibition. It is also a weak inhibitor of OATP1B1 (IC50 ∼ 66 μM) .
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