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DFP00173

Product Specifications

CAS Number

672286-03-2

Target

Aquaporin

Applications

Transmembrane Transporters

Molecular Formula

C11H7Cl2N3O3S

Additionnal Information

DFP00173 is a selective and potent inhibitor of Aquaporin-3 (AQP3), it inhibits mouse and human AQP3 with an IC50 of ∼0.1 μM–0.4 μM. It demonstrates potential for treating human disorders of water retention.

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