What is the catalog number for Pitolisant?

The catalog number for Pitolisant is E4955-100mg.

What sizes are available for Pitolisant?

Pitolisant is available in the following size(s): 100 mg.

Is Pitolisant in stock?

Pitolisant is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures Pitolisant?

Pitolisant is manufactured by Bimake.

What is the estimated delivery time for Pitolisant?

Estimated delivery time for Pitolisant is approximately 15 business day(s), depending on your location.

Pitolisant

Product Specifications

CAS Number

362665-56-3

Synonyms

BF2.649, Tiprolisant

Target

Histamine Receptor

Applications

Neuronal Signaling

Additionnal Information

Pitolisant (BF2.649, Tiprolisant) is a potent, selective antagonist of the non-imidazole histamine H3 receptor, with a Ki value of 0.16 nM and an EC50 of 1.5 nM as an inverse agonist. It enhances the activity of histaminergic neurons, promoting vigilance and cognitive function. It is useful in research on wakefulness, memory deficits, and cognitive disorders.