Teneligliptin Hydrobromide Hydrate

Product Specifications

CAS Number

1572583-29-9

Synonyms

MP-513 hydrobromide hydrate

Target

DPP

Applications

Metabolism

Molecular Formula

C22H30N6OS.5/2BrH.xH2O

Additionnal Information

Teneligliptin Hydrobromide Hydrate (MP-513 hydrobromide hydrate) is a potent, competitive, and long-lasting inhibitor of DPP-4. It competitively inhibited rhDPP-4, human plasma, and rat plasma with IC50 values of 0.889, 1.75, and 1.35 nM respectively. It suppresses high glucose-mediated mitochondrial dysfunction and can be used for treatment of type 2 diabetes.