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BML-284

Product Specifications

CAS Number

853220-52-7

Synonyms

Wnt Agonist

Target

Wnt/beta-catenin

Applications

Cytoskeletal Signaling

Molecular Formula

C19H18N4O3

Additionnal Information

BML-284 (Wnt Agonist) is a potent and cell-permeable activator of Wnt signaling that induces TCF-dependent transcriptional activity with an EC50 value of 0.7 μM. BML-284 also acts as an agonist of β-catenin that effectively activates direct Wnt-β-catenin signaling to induce adipocyte dedifferentiation while circumventing the apoptotic effect in the hypertonic treatment.

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