Oveporexton (TAK-861)
Product Specifications
CAS Number
2460722-04-5
Target
OX Receptor
Applications
Neuronal Signaling
Molecular Formula
C23H25F5N2O4S
Additionnal Information
Oveporexton (TAK-861) is a potent, orally bioavailable agonist of orexin receptor 2 (OX2R), with an EC50 of 2.5 nM in calcium mobilization assays. It induces dose-dependent membrane depolarization in histaminergic neurons within the mouse tuberomammillary nucleus (TMN) with an EC50 of 31.7 nM.
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