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BBC0403

Product Specifications

CAS Number

2644662-83-7

Target

Epigenetic Reader Domain

Applications

Epigenetics

Molecular Formula

C21H22N2O5

Additionnal Information

BBC0403 is a small-molecule selective inhibitor of Bromodomain-containing protein 2 (BRD2) with Kds of 7.64 μM and 41.37 μM for BRD2 (BD2) and BRD2 (BD1), respectively. It is a potential intra-articular injectable therapeutic agent for treating osteoarthritis (OA) .

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